2018
- From a Helix to a Small Cycle: Metadynamics-Inspired αvβ6 Integrin Selective Ligands
- In vivo characterization of four 68Ga-labeled multimeric RGD peptides to image αvβ3 integrin expression in two human tumor xenograft mouse models
- N-Methylation of isoDGR Peptides: Discovery of a Selective α5β1-Integrin Ligand as a Potent Tumor Imaging Agent
- Therapeutic Radiopharmaceuticals Targeting Integrin αvβ6
2016
- In-vivo PET imaging of the "cancer integrin" αvβ6 using gallium-68 labelled cyclic RGD nonapeptides
- Variation of Specific Activities of 68Ga-Aquibeprin and 68Ga-Avebetrin Enables Selective PET Imaging of Different Expression Levels of Integrins a5b1 and avb3
- Tailoring Fluorescent Dyes To Optimize a Hybrid RGD-Tracer
Ältere
- Comparison of cyclic RGD peptides for αvβ3 integrin detection in a rat model of myocardial infarction
- Be spoilt for choice with radiolabelled RGD peptides: Preclinical evaluation of 68 Ga-TRAP(RGD)3
- 68Ga-NODAGA-RGD is a suitable substitute for 18F-Galacto-RGD and can be produced with high specific activity in a cGMP/GRP compliant automated process