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Technische Universität München
  • Lehrstuhl für Pharmazeutische Radiochemie
  • TUM School of Natural Sciences
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  • Radiochemie München
Technische Universität München
  • Lehrstuhl für Pharmazeutische Radiochemie
  • TUM School of Natural Sciences
  • Technische Universität München
  1. Aktuelles
  2. Publikationen
  3. Integrine

2018

  • From a Helix to a Small Cycle: Metadynamics-Inspired αvβ6 Integrin Selective Ligands
  • In vivo characterization of four 68Ga-labeled multimeric RGD peptides to image αvβ3 integrin expression in two human tumor xenograft mouse models
  • N-Methylation of isoDGR Peptides: Discovery of a Selective α5β1-Integrin Ligand as a Potent Tumor Imaging Agent
  • Therapeutic Radiopharmaceuticals Targeting Integrin αvβ6

2017

  • A Comprehensive Evaluation of the Activity and Selectivity Profile of Ligands for RGD-binding Integrins

2016

  • In-vivo PET imaging of the "cancer integrin" αvβ6 using gallium-68 labelled cyclic RGD nonapeptides
  • Variation of Specific Activities of 68Ga-Aquibeprin and 68Ga-Avebetrin Enables Selective PET Imaging of Different Expression Levels of Integrins a5b1 and avb3
  • Tailoring Fluorescent Dyes To Optimize a Hybrid RGD-Tracer

2015

  • In vivo biokinetic and metabolic characterization of the 68Ga-labelled α5β1-selective peptidomimetic FR366

Ältere

  • Comparison of cyclic RGD peptides for αvβ3 integrin detection in a rat model of myocardial infarction
  • Be spoilt for choice with radiolabelled RGD peptides: Preclinical evaluation of 68 Ga-TRAP(RGD)3
  • 68Ga-NODAGA-RGD is a suitable substitute for 18F-Galacto-RGD and can be produced with high specific activity in a cGMP/GRP compliant automated process
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Lehrstuhl für Pharmazeutische Radiochemie

Prof. Dr. Angela Casini

Walther-Meißner-Str. 3
85748 Garching
Germany

Tel +49.89.289.12203
Fax +49.89.289.12204

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